![serotonin transporter serotonin transporter](https://image.slidesharecdn.com/review-130215120652-phpapp01/95/evidence-of-serotonin-transporter-gene-s-allele-being-a-plasticity-gene-2-638.jpg)
Clomipramine is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with K i of 0.14, 54 and 3 nM, respectively. Centanafadine hydrochloride is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC 50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter, respectively.Ĭhlorimipramine-d3 G-34586-d3 NSC-169865-d3Ĭlomipramine-d3 (Chlorimipramine-d3) is the deuterium labeled Clomipramine. HY-16736AS Centanafadine-d7 hydrochlorideĬentanafadine-d7 (EB-1020-d7) hydrochloride is the deuterium labeled Centanafadine hydrochloride.Indatraline hydrochloride may also serve to direct the development of new agents for autophagy-related diseases such as atherosclerosis or restenosis.Īdrenergic Receptor Dopamine Transporter Serotonin TransporterĬentanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC 50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter, respectively.Ĭentanafadine (hydrochloride) is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC 50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter, respectively. Indatraline hydrochloride induces autophagy while simultaneously inhibiting cell proliferation. Indatraline hydrochloride can be used for the research of antidepressive. Indatraline hydrochloride (Lu 19-005) is a non-selective monoamine transporter inhibitor that blocks the reuptake of neurotransmitters ( dopamine, serotonin, and norepinephrine) with efficacy similar to cocaine. Serotonin Transporter Dopamine Transporter